SCHEMBL4586422

SCHEMBL4586422

Cc1cc(-c2ccncc2)cc(C)c1C(=O)NC(C)CCN1CCC(N(Cc2ccccc2)c2ccc(C(=O)O)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.47
DRD2 P14416 2/20 0.44
DRD3 P35462 2/20 0.44
ROCK2 O75116 3/20 0.40
ROCK1 Q13464 2/20 0.40
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585297 0.87 CCR5 (0.48) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4586072 0.85 CCR5 (0.57) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4249206 0.84 CCR5 (0.68) CCR5
SCHEMBL4585280 0.83 CCR5 (0.48) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4586226 0.81 CCR5 (0.50) CCR5DRD2DRD3DCUN1D1
SCHEMBL4586504 0.81 CCR5 (0.56) CCR5DRD2DRD3
SCHEMBL4585572 0.79 CCR5 (0.52) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4240465 0.78 CCR5 (0.62) CCR5
SCHEMBL4586981 0.77 CCR5 (0.49) CCR5DRD2DRD3DCUN1D1
SCHEMBL4248706 0.77 CCR5 (0.74) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed