SCHEMBL4586633

SCHEMBL4586633

Brc1ccoc1-c1nc(N2CCNCC2)no1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.46
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HTR2C P28335 1/20 0.36
ADRB1 P08588 1/20 0.36
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2244692 0.76 ALDH1A1 (0.51) NPC1RAB9AADRB1
Hydrochloric Acid SCHEMBL2247573 0.74 ALDH1A1 (0.50) NPC1RAB9AADRB1
SCHEMBL11988503 0.74 ADRB2 (0.49) NPC1RAB9AHRH1
Hydrochloric Acid SCHEMBL2247082 0.73 ADRB2 (0.47) NPC1RAB9AHRH1
SCHEMBL4586732 0.71 MEN1 (0.45) NPC1RAB9AHTR2CHRH1
SCHEMBL30579597 0.69 NPC1 (0.41) NPC1RAB9AADRB1HRH1
SCHEMBL2248381 0.69 NPC1 (0.75) NPC1RAB9AADRB1
SCHEMBL9119904 0.67 HTR6 (0.46) HTR2CADRB1
SCHEMBL4585928 0.67 CASP3 (0.50) CASP3NPC1RAB9AHTR2C
SCHEMBL21938846 0.65 FEN1 (0.40) NPC1RAB9AHTR2CADRB1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581213-A4 3,5-DISUBSTITUTED- 1,2,4 -OXADIAZOLES AND ANALOGS AS AC TIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA INC (US) 2008-11-19 EP claimed
EP-1581213-A1 3,5-DISUBSTITUTED- 1,2,4 -OXADIAZOLES AND ANALOGS AS AC TIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF Cytovia, Inc. (US) 2005-10-05 EP claimed
WO-2004058253-A1 3,5-DISUBSTITUTED-[1,2,4]-OXADIAZOLES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2004-07-15 WO claimed