SCHEMBL4589758

SCHEMBL4589758

C=CCOC(=O)NCCc1cccc(Cl)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MTNR1A P48039 2/20 0.41
HPGD P15428 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
HIF1A Q16665 1/20 0.39
CNR1 P21554 1/20 0.39
CASP1 P29466 2/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
FAAH O00519 1/20 0.38
CYP3A4 P08684 1/20 0.38
NQO2 P16083 1/20 0.38
CTSG P08311 1/20 0.37
CMA1 P23946 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1821309 0.89 HIF1A (0.50) ERN1MEN1KMT2AHPGDALDH1A1
SCHEMBL4590421 0.76 ALDH1A1 (0.55) MEN1KMT2AHPGDALDH1A1TAAR1
SCHEMBL29168148 0.76 NQO2 (0.57) MEN1KMT2AHPGDALDH1A1CYP3A4
SCHEMBL4535306 0.75 HIF1A (0.51) MEN1KMT2ATAAR1HIF1ACNR1
SCHEMBL6999007 0.71 CASP1 (0.46) ERN1MEN1KMT2AALDH1A1CASP1
SCHEMBL20146223 0.71 ERN1 (0.47) ERN1MEN1KMT2AHPGDALDH1A1
SCHEMBL28259385 0.71 FAAH (0.65) MEN1KMT2AFAAHTRPV1CYP1A2
SCHEMBL13055388 0.71 MAPT (0.42) ERN1MEN1KMT2ACASP1CYP3A4
SCHEMBL807757 0.71 HIF1A (0.54) KMT2AHPGDALDH1A1TAAR1HIF1A
SCHEMBL15468130 0.71 HIF1A (0.54) KMT2AHPGDALDH1A1TAAR1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937656-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS BETA 2 ADRENOCEPTOR AGONISTS AstraZeneca AB (SE) 2008-07-02 EP disclosed
WO-2007027134-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS β2 ADRENOCEPTOR AGONISTS ASTRAZENECA AB (SE) 2007-03-08 WO disclosed