SCHEMBL4592244

SCHEMBL4592244

OC(=S)Cc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTBP2 P56545 1/20 0.48
ALDH1A1 P00352 2/20 0.47
FAAH O00519 1/20 0.47
MGLL Q99685 1/20 0.47
L3MBTL1 Q9Y468 3/20 0.45
MAPT P10636 2/20 0.45
TDP1 Q9NUW8 1/20 0.44
IDO1 P14902 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
HPGD P15428 2/20 0.43
ALOX12 P18054 1/20 0.43
LMNA P02545 1/20 0.42
PIK3CA P42336 2/20 0.41
CNR2 P34972 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPK1 P28482 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11539903 0.88 MAPT (0.45) CTBP2ALDH1A1FAAHMGLLL3MBTL1
SCHEMBL11537202 0.88 LTA4H (0.50) CTBP2ALDH1A1FAAHMGLLMAPT
SCHEMBL11084515 0.80 CA2 (0.41) CTBP2ALDH1A1FAAHMGLLMAPT
SCHEMBL10610797 0.80 ALDH1A1 (0.47) CTBP2ALDH1A1FAAHMGLLL3MBTL1
SCHEMBL1999167 0.78 IDO1 (0.52) CTBP2ALDH1A1FAAHMGLLL3MBTL1
SCHEMBL11081484 0.77 TSHR (0.50) TDP1LMNA
SCHEMBL10524113 0.77 CA2 (0.58) CTBP2ALDH1A1L3MBTL1MAPTTDP1
SCHEMBL28210144 0.76 IDO1 (0.50) IDO1MEN1KMT2ATAAR1
SCHEMBL4066362 0.76 L3MBTL1 (0.52) CTBP2ALDH1A1L3MBTL1MAPTTDP1
SCHEMBL1096270 0.76 CES1 (0.55) CTBP2ALDH1A1L3MBTL1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118496175-A TRADD inhibitor derivative and preparation method and application thereof 安徽医科大学 2024-08-16 CN claimed
CN-118496175-A TRADD inhibitor derivative and preparation method and application thereof 安徽医科大学 2024-08-16 CN disclosed
US-11932653-B2 Lycorine derivative, and pharmaceutical composition and use thereof SHANDONG DYNE MARINE BIOPHARMACEUTICAL CO., LTD (CN) 2024-03-19 US disclosed
US-20210206777-A1 LYCORINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF SHANDONG DYNE MARINE BIOPHARMACEUTICAL CO., LTD (CN) 2021-07-08 US disclosed
CN-107722049-B Preparation and application of novel ionic binuclear Schiff base titanium complex 山西医科大学 2020-06-30 CN disclosed
WO-2020019357-A1 LYCORINE DERIVATIVES, PHARMACEUTICAL COMPOSITE THEREOF AND USAGE THEREFOR 山东达因海洋生物制药股份有限公司 2020-01-30 WO disclosed
US-7442485-B2 Lithographic process involving on press development FUJIFILM CORPORATION (JP) 2008-10-28 US disclosed
EP-1484177-B1 Lithographic process involving on press development FUJIFILM CORP (JP) 2007-08-29 EP disclosed
US-20050016402-A1 Lithographic process involving on press development FUJI PHOTO FILM CO., LTD. 2005-01-27 US disclosed
EP-1484177-A2 Lithographic process involving on press development FUJI PHOTO FILM CO., LTD. (JP) 2004-12-08 EP disclosed
EP-0207690-B1 N-SUBSTITUTED GLUTAMIC ACID DERIVATIVE AND PROCESS FOR PRODUCTION AND USE THEREOF SUNTORY LIMITED (JP) 1989-12-20 EP disclosed
EP-0146297-B1 SUBSTITUTED TRANS-1,2-DIAMINOCYCLOHEXYL AMIDE COMPOUNDS WARNER-LAMBERT COMPANY (US) 1988-02-03 EP disclosed
US-4701210-A HERBICIDES SUNTORY LIMITED (JP) 1987-10-20 US disclosed
US-4677122-A ANALGESICS, DIURETICS WARNER-LAMBERT COMPANY (US) 1987-06-30 US disclosed
EP-0207690-A1 N-Substituted glutamic acid derivative and process for production and use thereof SUNTORY LIMITED (JP) 1987-01-07 EP disclosed
US-4598087-A DIURETICS; ANALGESICS, PSYCHOTHERAPEUTICS WARNER-LAMBERT COMPANY (US) 1986-07-01 US disclosed
EP-0146297-A1 Substituted trans-1,2-diaminocyclohexyl amide compounds WARNER-LAMBERT COMPANY (US) 1985-06-26 EP disclosed
EP-0027895-A1 1-(2-(Alkyl and arylsulfonyl)-2-propenyl and propyl) substituted piperidines and pharmaceutical and antimicrobial compositions comprising the same MERCK & CO. INC. (US) 1981-05-06 EP disclosed
US-4244963-A 1-[2-(Alkyl and arylsulfonyl)-2-propenyl and propyl] substituted piperidines useful as antimicrobial and antiinflammatory agents MERCK & CO., INC. (US) 1981-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11932653-B2 Lycorine derivative, and pharmaceutical composition and use thereof LCT, LARP7, LASP1 CTBP2 4530/4885ALDH1A1 2939/4885FAAH 3663/4885
US-20210206777-A1 LYCORINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF LARP7, LARP1, LASP1 CTBP2 4476/4885ALDH1A1 2613/4885FAAH 3958/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.