SCHEMBL4592830

SCHEMBL4592830

CS(=O)(=O)c1nc(OCc2ccccc2)cc(-c2cccc(C(F)(F)F)c2)n1.N#Cc1nc(OCc2ccccc2)cc(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 17/20 0.50
CTSS P25774 5/20 0.50
KCNH2 Q12809 14/20 0.46
CTSB P07858 4/20 0.45
CTSL P07711 3/20 0.45
SDHB P21912 2/20 0.44
MEN1 O00255 1/20 0.43
S1PR4 O95977 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
S1PR1 P21453 1/20 0.43
MAPK1 P28482 1/20 0.43
STAT3 P40763 1/20 0.43
STAT1 P42224 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3875432 0.92 SDHB (0.51) KCNH2SDHBMEN1S1PR4LMNA
SCHEMBL3873029 0.90 CTSK (0.57) CTSKCTSSKCNH2CTSBCTSL
SCHEMBL14267874 0.77 SQOR (0.59) CTSKCTSSMAPK1RAB9A
SCHEMBL5593061 0.76 SDHB (0.68) SDHBMEN1S1PR4LMNATP53
SCHEMBL3875774 0.74 LMNA (0.46) CTSKCTSSLMNAHPGDHSD17B10
SCHEMBL3874622 0.73 CTSK (0.60) CTSKCTSSKCNH2CTSBCTSL
SCHEMBL8560362 0.73 SDHB (0.56) SDHBMEN1S1PR4LMNATP53
SCHEMBL3877426 0.72 CTSK (0.68) CTSKCTSSKCNH2CTSBCTSL
SCHEMBL27739899 0.72 PTPN1 (0.42) CTSKCTSSMEN1KMT2A
SCHEMBL19805611 0.72 SDHB (0.74) KCNH2SDHBMEN1S1PR4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928842-A1 4-PHENYL-6-SUBSTITUTED-PYRIMIDINE-2-CARBONITRILE DERIVATIVES N.V. Organon (NL) 2008-06-11 EP disclosed
WO-2007039470-A1 4-PHENYL-6-SUBSTITUTED-PYRIMIDINE-2-CARBONITRILE DERIVATIVES N.V. ORGANON (NL) 2007-04-12 WO disclosed