SCHEMBL4593299

SCHEMBL4593299

COc1ccc(C2(C(Cl)(Cl)C3(c4ccc(OC)cc4)N=NN=N3)N=NN=N2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
MAPK1 P28482 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
TSHR P16473 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA12 O43570 1/20 0.42
CA14 Q9ULX7 1/20 0.42
MAOB P27338 2/20 0.38
MAOA P21397 1/20 0.38
ACHE P22303 1/20 0.37
IDO1 P14902 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
MAPT P10636 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5298336 0.74 CA1 (0.48) ALDH1A1MAPK1TDP1L3MBTL1CA1
SCHEMBL4593190 0.74 SLC6A3 (0.33) MAOBMAOAIDO1
SCHEMBL10765712 0.72 CA1 (0.46) ALDH1A1MAPK1TDP1L3MBTL1CA1
SCHEMBL5287713 0.68 HSD11B1 (0.51) ALDH1A1MAPK1L3MBTL1CA1CA2
SCHEMBL2007523 0.66 KCNQ3 (0.39) ALDH1A1MAPK1TSHRL3MBTL1MEN1
SCHEMBL5301951 0.66 CES2 (0.41) MAPK1CA1CA2CA7CA9
1,4-Dimethoxybenzene SCHEMBL8489 0.65 CA1 (1.00) ALDH1A1MAPK1TDP1L3MBTL1CA1
1,4-Dimethoxybenzene SCHEMBL21802643 0.65 CA1 (1.00) ALDH1A1MAPK1TDP1L3MBTL1CA1
SCHEMBL10642557 0.63 CA1 (0.58) ALDH1A1MAPK1TDP1TSHRL3MBTL1
SCHEMBL11470325 0.63 CA1 (0.58) ALDH1A1MAPK1TDP1TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP claimed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO claimed
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP disclosed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO disclosed