SCHEMBL4593445

SCHEMBL4593445

Cc1ccccc1C1(C(Cl)C2(c3ccccc3C)N=NN=N2)N=NN=N1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.34
TSHR P16473 1/20 0.33
ACHE P22303 1/20 0.33
CYP3A4 P08684 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
OPRM1 P35372 2/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
OPRL1 P41146 1/20 0.31
CD44 P16070 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8705403 0.69 TSHR (0.38) HDAC4TSHRACHECYP3A4TDP1
SCHEMBL4593516 0.68 ACHE (0.33) ACHETDP1
SCHEMBL11470022 0.63 ACHE (0.45) HDAC4TSHRACHECYP3A4TDP1
O-Xylene SCHEMBL2858075 0.63 TSHR (0.71) TSHRACHECYP3A4TDP1
O-Xylene SCHEMBL2589554 0.61 TSHR (0.67) TSHRACHECYP3A4TDP1
O-Xylene SCHEMBL10353038 0.61 TSHR (0.67) TSHRACHECYP3A4TDP1
SCHEMBL19743353 0.60 PDK2 (0.43) TSHRACHECYP3A4TDP1
O-Xylene SCHEMBL5375995 0.59
SCHEMBL8984654 0.57 ESR1 (0.50) HDAC4TSHRACHECYP3A4TDP1
SCHEMBL6351769 0.57 ESR1 (0.50) TSHRACHECYP3A4TDP1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP claimed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO claimed
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP disclosed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO disclosed