SCHEMBL4593796

SCHEMBL4593796

Cc1ccc(C)n1-c1cc(CO)ccn1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.47
VHL P40337 1/20 0.39
MAOA P21397 1/20 0.38
DYRK1A Q13627 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
ALDH1A1 P00352 4/20 0.36
LMNA P02545 3/20 0.36
SORD Q00796 4/20 0.36
KDM4E B2RXH2 3/20 0.36
KLKB1 P03952 1/20 0.35
CTSB P07858 1/20 0.35
KDM5A P29375 2/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
MAPT P10636 1/20 0.34
KDM4C Q9H3R0 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PLAU P00749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13040670 0.86 ALDH1A1 (0.35) RECQLALDH1A1LMNASORDKDM4E
SCHEMBL18585998 0.82 ALDH1A1 (0.36) ALDH1A1LMNAKDM4EKDM5ALOXL2
SCHEMBL13040657 0.81 ALDH1A1 (0.36) RECQLALDH1A1LMNAKDM4EKDM5A
SCHEMBL18586168 0.79 KLKB1 (0.38) ALDH1A1LMNASORDKDM4EKLKB1
SCHEMBL4334724 0.78 KDM4E (0.41) ALDH1A1LMNAKDM4ELOXL2L3MBTL1
Propanol SCHEMBL6771763 0.76 ALDH1A1 (0.48) RECQLALDH1A1LMNAKDM4EL3MBTL1
SCHEMBL6619720 0.75 ALDH1A1 (0.57) RECQLALDH1A1LMNAKDM4EL3MBTL1
SCHEMBL17781654 0.74 RECQL (0.50) RECQLVHLMAOADYRK1AHRH3
SCHEMBL22898276 0.74 SORD (0.53) RECQLHRH3SORD
SCHEMBL4594579 0.73 AKT1 (0.36) HRH3ALDH1A1LMNAKDM5AKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891047-A4 1-METHYL-1H-PYRAZOLE-4-CARBOXAMIDES USEFUL AS CANCER CHEMOTHERAPEUTIC AGENTS BAYER HEALTHCARE AG (DE) 2008-07-09 EP disclosed
EP-1891047-A2 1-METHYL-1H-PYRAZOLE-4-CARBOXAMIDES USEFUL AS CANCER CHEMOTHERAPEUTIC AGENTS Bayer HealthCare AG (DE) 2008-02-27 EP disclosed
WO-2006133006-A2 1-METHYL-1H-PYRAZOLE-4-CARBOXAMIDES USEFUL AS CANCER CHEMOTHERAPEUTIC AGENTS BAYER HEALTHCARE AG (DE) 2006-12-14 WO disclosed