SCHEMBL4595113

SCHEMBL4595113

[CH2]C1Cc2cccc(Nc3ccc(Cl)cc3)c2O1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.35
TRPV1 Q8NER1 1/20 0.34
MAPK14 Q16539 1/20 0.33
LMNA P02545 2/20 0.33
SHMT2 P34897 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
PKM P14618 1/20 0.32
KDM4E B2RXH2 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
MPI P34949 1/20 0.32
NFKB1 P19838 2/20 0.31
NFKB2 Q00653 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596760 0.86 MAPT (0.43) POLBMAPK14LMNAKDM4ECYP1A2
SCHEMBL4595116 0.82 PARP1 (0.44) POLBTRPV1MAPK14NPSR1PKM
SCHEMBL4230647 0.79 AQP1 (0.43) POLBTRPV1MAPK14LMNASHMT2
SCHEMBL4711112 0.72 HTR2A (0.36) MAPK14NPSR1MAPTALDH1A1HTT
SCHEMBL4595476 0.70 L3MBTL1 (0.35) POLBLMNAKDM4EHPGDALDH1A1
SCHEMBL4595291 0.70 AQP1 (0.44) MAPK14NPSR1KDM4ECYP1A2MAPT
SCHEMBL4597588 0.69 HTR7 (0.43)
SCHEMBL4595494 0.69 AQP1 (0.36)
SCHEMBL4233314 0.69 PRKAB2 (0.44) SHMT2
SCHEMBL4222627 0.68 PRKAB2 (0.43) POLBMAPTHPGDKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed