SCHEMBL4595429

SCHEMBL4595429

Fc1cccc(-c2cc(Cl)cc3c2OC([CH]Cc2ccccc2)C3)c1F

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596984 0.81 AQP1 (0.45) AQP1SIRT2HTR2AHTR2C
SCHEMBL4596492 0.81 AQP1 (0.36) AQP1SIRT2HTR2AHTR2C
SCHEMBL4595432 0.80 SIRT2 (0.52) AQP1SIRT2HTR2A
SCHEMBL4595082 0.79 AQP1 (0.33) AQP1SIRT2
SCHEMBL4596725 0.77 CHRM1 (0.33) AQP1SIRT2
SCHEMBL4596675 0.76 AQP1 (0.37) AQP1SIRT2
SCHEMBL4596587 0.76 HTR2A (0.37) AQP1HTR2AHTR2C
SCHEMBL4596590 0.76 HTR1A (0.38) AQP1HTR2AHTR2C
SCHEMBL4220557 0.75 AQP1 (0.56) AQP1SIRT2HTR2AHTR2C
SCHEMBL4596775 0.75 AQP1 (0.40) AQP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed