SCHEMBL4596775

SCHEMBL4596775

Clc1ccc(-c2cccc3c2OC([CH]Cc2ccccc2)C3)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 2/20 0.40
CYP1A2 P05177 2/20 0.36
NPC1 O15118 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DPP4 P27487 1/20 0.35
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
GRM5 P41594 1/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596725 0.91 CHRM1 (0.33) AQP1CYP1A2NPC1CYP2C19RAB9A
SCHEMBL4596399 0.89 HTR1A (0.34) AQP1L3MBTL1ALDH1A1NPSR1MEN1
SCHEMBL4596984 0.89 AQP1 (0.45) AQP1CYP1A2NPC1CYP2D6CYP2C9
SCHEMBL4595082 0.88 AQP1 (0.33) AQP1DPP4SLC6A2SLC6A4MEN1
SCHEMBL4596103 0.86 AQP1 (0.43) AQP1CYP1A2NPC1CYP2D6CYP2C9
SCHEMBL6047944 0.85 P2RX7 (0.38) L3MBTL1SLC6A2SLC6A4
SCHEMBL4596675 0.83 AQP1 (0.37) AQP1L3MBTL1
SCHEMBL6047967 0.80 MAPK1 (0.33) NPC1RAB9ASMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL4596928 0.80 PRKAB2 (0.35) SMN1; SMN2ALDH1A1MAPT
SCHEMBL4596777 0.78 SIRT2 (0.49) AQP1CYP1A2NPC1CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed