SCHEMBL4596005

SCHEMBL4596005

COc1cccc(-c2cccc3c2OC([CH]Cc2ccccc2)C3)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.42
TMEM97 Q5BJF2 3/20 0.42
SIGMAR1 Q99720 3/20 0.42
DRD4 P21917 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
SLC6A3 Q01959 2/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
OPRK1 P41145 1/20 0.42
HTR5A P47898 1/20 0.42
PRKAB2 O43741 1/20 0.41
PRKAG1 P54619 1/20 0.41
PRKAA2 P54646 1/20 0.41
PRKAA1 Q13131 1/20 0.41
PRKAG3 Q9UGI9 1/20 0.41
PRKAG2 Q9UGJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596329 0.85 CYP1A1 (0.40) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4596532 0.79 PRKAB2 (0.40) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4596007 0.79 PRKAB2 (0.49) HTR1ATMEM97SIGMAR1DRD4HTR2C
SCHEMBL6047967 0.78 MAPK1 (0.33) HTR2CPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4597055 0.76 HTR1A (0.49) HTR1APRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4596399 0.76 HTR1A (0.34) HTR1ADRD4HTR2CHTR7DRD3
SCHEMBL4597054 0.75 HTR1A (0.48) HTR1APRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4595082 0.75 AQP1 (0.33) SLC6A2SLC6A4PRKAB2PRKAG1PRKAA2
SCHEMBL4596675 0.75 AQP1 (0.37) DRD4DRD3
SCHEMBL4220641 0.75 PRKAB2 (0.69) HTR1APRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
WO-2007030150-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH (US) 2007-03-15 WO disclosed