SCHEMBL4597474

SCHEMBL4597474

CON1c2ccc(C(=O)N3CCNCC3)cc2C(C)(C)[C@H]2COc3ccccc3[C@H]21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.37
PDE4B Q07343 1/20 0.36
MEN1 O00255 2/20 0.35
USP2 O75604 2/20 0.35
KMT2A Q03164 2/20 0.35
TSHR P16473 1/20 0.35
CNR2 P34972 2/20 0.34
KDR P35968 1/20 0.34
HPGD P15428 2/20 0.34
LMNA P02545 1/20 0.34
HSD11B1 P28845 2/20 0.33
HCRTR2 O43614 1/20 0.33
CHRM3 P20309 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598721 0.88 PDE4B (0.39) SIGMAR1PDE4BMEN1USP2KMT2A
SCHEMBL4563416 0.85 LTB4R (0.36) TSHRHCRTR2
SCHEMBL4564083 0.84 TSHR (0.42) MEN1KMT2ATSHRHCRTR2
SCHEMBL4628825 0.80 RARB (0.39) PDE4BHCRTR2
SCHEMBL4564105 0.79 PDE4A (0.37) PDE4BMEN1KMT2ATSHRHCRTR2
SCHEMBL4447404 0.79 DRD2 (0.40)
SCHEMBL4564085 0.77 HSP90AA1 (0.39) MEN1KMT2AHSD11B1
SCHEMBL4629499 0.77 HSP90AA1 (0.39) KMT2ALMNA
SCHEMBL4566254 0.76 PDK2 (0.41) MEN1KMT2A
SCHEMBL4566136 0.76 PDK2 (0.41) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907395-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-04-09 EP disclosed
WO-2007002867-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2007-01-04 WO disclosed