SCHEMBL4447404

SCHEMBL4447404

CON1c2ccc(C(=O)NCCO)cc2C(C)(C)[C@H]2COc3ccccc3[C@H]21

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.40
DRD3 P35462 12/20 0.40
FSHR P23945 1/20 0.39
HTR2B P41595 1/20 0.38
GNRHR P30968 2/20 0.36
POLB P06746 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4563416 0.85 LTB4R (0.36) HTR2BALDH1A1
SCHEMBL4564083 0.84 TSHR (0.42) HTR2BALDH1A1
SCHEMBL4628825 0.80 RARB (0.39) FSHR
SCHEMBL4564105 0.79 PDE4A (0.37) FSHRHTR2B
SCHEMBL4598844 0.79 HCRTR1 (0.34) HTR2BALDH1A1
SCHEMBL4597474 0.79 SIGMAR1 (0.37)
SCHEMBL4566254 0.78 PDK2 (0.41)
SCHEMBL4566136 0.78 PDK2 (0.41)
SCHEMBL4565660 0.78 PDK2 (0.41) FSHRNPC1RAB9A
SCHEMBL4629499 0.77 HSP90AA1 (0.39) DRD2DRD3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125825-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2009-12-02 EP disclosed
WO-2008079139-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-07-03 WO disclosed