SCHEMBL4597590

SCHEMBL4597590

CC1Cc2cccc(-c3cc(Cl)cc(Cl)c3)c2O1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.46
HTR7 P34969 2/20 0.46
PARP1 P09874 3/20 0.46
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
PRKAB2 O43741 2/20 0.38
PRKAG1 P54619 2/20 0.38
PRKAA2 P54646 2/20 0.38
PRKAA1 Q13131 2/20 0.38
PRKAG3 Q9UGI9 2/20 0.38
PRKAG2 Q9UGJ0 2/20 0.38
PRKAB1 Q9Y478 2/20 0.38
BRD4 O60885 5/20 0.38
CREBBP Q92793 5/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595495 0.85 PARP1 (0.46) HTR1AHTR7PARP1MAOAMAOB
SCHEMBL4597588 0.82 HTR7 (0.43) HTR1AHTR7PRKAB2PRKAG1PRKAA2
SCHEMBL4596981 0.81 PARP1 (0.48) HTR1AHTR7PARP1MAOAMAOB
SCHEMBL4596910 0.80 PARP1 (0.49) HTR1AHTR7PARP1MAOAMAOB
SCHEMBL4712948 0.79 BRD4 (0.44) HTR1APARP1MAOAMAOBBRD4
SCHEMBL4595292 0.79 AQP1 (0.44) HTR1AHTR7PARP1MAOAMAOB
SCHEMBL4225611 0.78 PRKAB2 (0.62) HTR1AHTR7MAOBPRKAB2PRKAG1
SCHEMBL4595480 0.78 PARP1 (0.43) HTR1APARP1MAOAMAOBPRKAB2
SCHEMBL4595395 0.78 PARP1 (0.43) HTR1APARP1MAOAMAOBPRKAB2
SCHEMBL4649844 0.78 PARP1 (0.48) HTR1AHTR7PARP1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed