SCHEMBL4597735

SCHEMBL4597735

CN(C)C(=O)C(CNC(=O)OC(C)(C)C)c1ccc(Oc2ccc(CCC(N)=O)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.36
CA1 P00915 5/20 0.36
FFAR1 O14842 3/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
SYK P43405 1/20 0.34
CA12 O43570 3/20 0.33
CA9 Q16790 3/20 0.33
ACACB O00763 2/20 0.33
ACACA Q13085 2/20 0.33
MMP13 P45452 1/20 0.33
PTGER4 P35408 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
PLAAT3 P53816 1/20 0.33
PLAAT5 Q96KN8 1/20 0.33
PLAAT2 Q9NWW9 1/20 0.33
PLAAT4 Q9UL19 1/20 0.33
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597234 0.92 NR1H2 (0.40) CA2CA1NR1H2NR1H3SYK
SCHEMBL4597275 0.89 MMP13 (0.37) CA2CA1SYKMMP13ALDH1A1
SCHEMBL5307198 0.85 SYK (0.41) FFAR1SYKACACBMMP13PLAAT3
SCHEMBL4607919 0.84 CTSS (0.41) CA2FFAR1NR1H2NR1H3ACACB
SCHEMBL4598537 0.81 GHSR (0.38) CA2CA1SYKCA12CA9
SCHEMBL4597428 0.81 HDAC2 (0.43) CA2CA1NR1H2SYKPTGER4
SCHEMBL4597733 0.80 ITGB3 (0.45) CA2MMP13
SCHEMBL14021684 0.80 ITGB3 (0.45) CA2MMP13
SCHEMBL1932821 0.77 SYK (0.47) CA1SYKCA12
SCHEMBL14021742 0.76 FFAR1 (0.42) FFAR1ACACBACACAALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907352-A2 NOVEL DERIVATIVES OF AMINO ACIDS FOR TREATMENT OF OBESITY AND RELATED DISORDERS Bexel Pharmaceuticals Inc (US) 2008-04-09 EP disclosed
WO-2007005774-A2 NOVEL DERIVATIVES OF AMINO ACIDS FOR TREATMENT OF OBESITY AND RELATED DISORDERS BEXEL PHARMACEUTICALS, INC. (US) 2007-01-11 WO disclosed