SCHEMBL4598537

SCHEMBL4598537

CN(C)C(=O)C(CNC(=O)OC(C)(C)C)c1ccc(Oc2ccc(C=O)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.38
ALDH1A1 P00352 2/20 0.36
PARP10 Q53GL7 1/20 0.36
PARP3 Q9Y6F1 1/20 0.36
KDM4E B2RXH2 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
MMP13 P45452 2/20 0.35
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
SYK P43405 1/20 0.34
CA12 O43570 3/20 0.33
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 3/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
AAK1 Q2M2I8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597735 0.81 CA2 (0.36) ALDH1A1MMP13SYKCA12CA1
SCHEMBL4597275 0.81 MMP13 (0.37) ALDH1A1MMP13SYKCA1CA2
SCHEMBL1932821 0.80 SYK (0.47) MAPTSYKCA12CA1CTSS
SCHEMBL6830538 0.76 NPC1 (0.44) ALDH1A1KDM4ENPC1MMP13ADRB2
SCHEMBL14003045 0.76 ITGB3 (0.47) MMP13CTSSCTSK
SCHEMBL4598533 0.76 ITGB3 (0.47) MMP13CTSSCTSK
SCHEMBL6830761 0.76 PTPRB (0.44) CA1CA2
SCHEMBL4597927 0.76 GRN (0.42) POLB
SCHEMBL12987768 0.75 ADRB2 (0.40) ALDH1A1KDM4ENPC1MAPTRAB9A
SCHEMBL4597564 0.75 MMP13 (0.36) MMP13ADRB2ADRB1SYKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1906731-A2 NOVEL HYDROXAMIC ACID-CONTAINING AMINO ACID DERIVATIVES Bexel Pharmaceuticals Inc (US) 2008-04-09 EP disclosed
WO-2007005603-A2 NOVEL HYDROXAMIC ACID-CONTAINING AMINO ACID DERIVATIVES BEXEL PHARMACEUTICALS, INC. (US) 2007-01-11 WO disclosed