SCHEMBL4597890

SCHEMBL4597890

NCc1ccc(CN2CCC(C3COCCC3(c3ccccc3)N3CCNC3=O)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 7/20 0.39
CHRM1 P11229 1/20 0.36
CHRM3 P20309 6/20 0.36
CHRM2 P08172 5/20 0.36
ACHE P22303 1/20 0.36
NCF1 P14598 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597761 0.88 KCNJ1 (0.44) CHRM3CHRM2ACHE
SCHEMBL4596620 0.87 NPSR1 (0.38) CXCR3CHRM3CHRM2
SCHEMBL4597887 0.69 CHRM3 (0.42) CXCR3CHRM3CHRM2NCF1
Benzylamine SCHEMBL27789840 0.63 NCF1 (0.78) NCF1
SCHEMBL113089 0.61 NCF1 (0.74) NCF1
SCHEMBL8775737 0.60 MEN1 (0.74) ACHE
SCHEMBL3063295 0.60 CHRM3 (0.59) CHRM3CHRM2ACHE
SCHEMBL18458216 0.59 SIGMAR1 (0.48) ACHENCF1
SCHEMBL8129380 0.59 ALDH1A1 (0.69) NCF1
Hydrochloric Acid SCHEMBL7985714 0.59 MEN1 (0.72) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed