SCHEMBL4597887

SCHEMBL4597887

NCc1ccc(CN2CCC(N3C(=O)NC[C@]3(c3ccccc3)C3CCOCC3)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 12/20 0.42
CHRM2 P08172 11/20 0.42
CXCR3 P49682 4/20 0.41
NCF1 P14598 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597759 0.88 KCNJ1 (0.51)
SCHEMBL4596616 0.86 CHRM3 (0.41) CHRM3CHRM2CXCR3
SCHEMBL4597403 0.79 CCR5 (0.52) CHRM3CHRM2CXCR3
SCHEMBL4596041 0.78 KDM4E (0.32) CHRM3
SCHEMBL4597256 0.71 DRD2 (0.34) CXCR3
SCHEMBL5181129 0.71 CXCR3 (0.48) CHRM3CHRM2CXCR3
SCHEMBL4596625 0.69 HTR2C (0.35) CHRM3CHRM2
SCHEMBL4597890 0.69 CXCR3 (0.39) CHRM3CHRM2CXCR3NCF1
Benzylamine SCHEMBL27789840 0.68 NCF1 (0.78) NCF1
SCHEMBL5572519 0.67 CCR5 (0.72) CHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed