SCHEMBL4598150

SCHEMBL4598150

CN(c1ccc2[nH]nnc2c1)c1c(NCc2cccc(O)c2)c(=O)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 2/20 0.45
MAP4K4 O95819 2/20 0.45
AKT2 P31751 2/20 0.45
PIM3 Q86V86 2/20 0.45
PBK Q96KB5 2/20 0.45
DCLK1 O15075 1/20 0.45
PHKG2 P15735 1/20 0.45
IRAK4 Q9NWZ3 1/20 0.45
PIM2 Q9P1W9 1/20 0.45
ROCK2 O75116 3/20 0.35
CDK1 P06493 2/20 0.35
MAPK1 P28482 2/20 0.35
ROCK1 Q13464 2/20 0.35
RPS6KB1 P23443 2/20 0.35
AURKB Q96GD4 2/20 0.35
PLK4 O00444 1/20 0.35
CHEK1 O14757 1/20 0.35
DAPK3 O43293 1/20 0.35
DYRK3 O43781 1/20 0.35
JAK2 O60674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598143 0.83 SRC (0.41) PRKD3MAP4K4AKT2PIM3PBK
SCHEMBL4900221 0.74 MAPKAPK2 (0.47) PRKD3MAP4K4AKT2PIM3PBK
SCHEMBL4897972 0.74 MAPKAPK2 (0.47) PRKD3MAP4K4AKT2PIM3PBK
SCHEMBL1229059 0.68 ROCK2 (0.49) PRKD3MAP4K4AKT2PIM3PBK
SCHEMBL1228817 0.67 JAK2 (0.34) PRKD3MAP4K4AKT2PIM3PBK
SCHEMBL4898767 0.66 RPS6KB1 (0.40) PRKD3MAP4K4AKT2PIM3PBK
SCHEMBL4598151 0.64 OPRK1 (0.38) AKT2ROCK2ROCK1RPS6KB1AURKB
SCHEMBL4598401 0.63 KDR (0.47) RPS6KB1AURKBKDRMAPTNLRP3
SCHEMBL10806200 0.63 TERT (0.48) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL4908137 0.63 ROCK1 (0.52) PRKD3MAP4K4AKT2PIM3PBK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed