SCHEMBL4598598

SCHEMBL4598598

CC(C)(C)NC(=O)C(NC(=O)O)c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 11/20 0.49
S1PR1 P21453 5/20 0.49
S1PR4 O95977 4/20 0.49
S1PR2 O95136 3/20 0.49
S1PR5 Q9H228 1/20 0.42
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
SLC6A2 P23975 2/20 0.42
CHRNA1 P02708 1/20 0.42
CHRNG P07510 1/20 0.42
ITGA5 P08648 1/20 0.42
CHRNB1 P11230 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
SLC6A4 P31645 1/20 0.42
CHRNA3 P32297 1/20 0.42
CYP2C19 P33261 1/20 0.42
HRH1 P35367 1/20 0.42
CHRNA7 P36544 1/20 0.42
OPRK1 P41145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5575575 0.84 S1PR3 (0.57) S1PR3S1PR1S1PR4S1PR2SLC6A2
SCHEMBL9640678 0.81 GLS (0.48) S1PR3S1PR1S1PR4S1PR2SLC6A2
SCHEMBL5573778 0.78 ROCK2 (0.46) S1PR3S1PR1S1PR4S1PR2SLC6A2
SCHEMBL6719076 0.73 MAPT (0.56) ALDH1A1SMN1; SMN2
SCHEMBL4595463 0.73 ADRB3 (0.44) CYP2C19
SCHEMBL4371128 0.72 TRPM8 (0.41) S1PR3S1PR1S1PR4S1PR2SLC6A2
SCHEMBL25342655 0.72 CNR1 (0.45) S1PR3S1PR4CYP2C19ALDH1A1
SCHEMBL25342652 0.72 CNR1 (0.45) S1PR3S1PR4CYP2C19ALDH1A1
SCHEMBL31749408 0.72 S1PR3 (0.58) S1PR3S1PR1S1PR4S1PR2
SCHEMBL15226465 0.72 MEN1 (0.45) ALDH1A1SMN1; SMN2ACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed