SCHEMBL4599900

SCHEMBL4599900

O=C(O)c1ccc(Oc2ncccc2C(=O)Nc2ccccc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.70
ALDH1A1 P00352 3/20 0.60
PPARG P37231 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56
NCOR2 Q9Y618 1/20 0.56
MAPK8 P45983 2/20 0.55
TDP1 Q9NUW8 1/20 0.54
NPC1 O15118 1/20 0.54
TP53 P04637 1/20 0.54
RECQL P46063 1/20 0.54
RAB9A P51151 1/20 0.54
GAA P10253 2/20 0.54
POLB P06746 1/20 0.54
PRKCI P41743 1/20 0.53
MEN1 O00255 1/20 0.52
MAPT P10636 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4939060 0.91 KMT2A (0.82) KMT2AALDH1A1MAPK8TDP1GAA
SCHEMBL4600567 0.90 KMT2A (0.82) KMT2AALDH1A1PPARGRXFP1NCOR2
SCHEMBL4599856 0.88 KMT2A (0.65) KMT2APPARGRXFP1NCOR2NPC1
SCHEMBL11810048 0.83 PDE10A (0.60) KMT2AALDH1A1MAPK8TDP1RAB9A
SCHEMBL2485533 0.83 KMT2A (0.67) KMT2A
SCHEMBL6120093 0.80 RAB9A (0.72) ALDH1A1MAPK8TDP1RAB9AGAA
SCHEMBL10973818 0.79 KMT2A (0.68) KMT2AALDH1A1PPARGRXFP1NCOR2
SCHEMBL10971064 0.79 ALDH1A1 (0.72) KMT2AALDH1A1MAPK8TDP1NPC1
SCHEMBL7906081 0.79 PDE10A (0.67) KMT2AALDH1A1TDP1
SCHEMBL14284685 0.77 PNLIP (0.68) KMT2AALDH1A1TDP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910295-A1 SUBSTITUTED PYRIDOCARBOXAMIDES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR 1 (PAI-1) Bayer HealthCare AG (DE) 2008-04-16 EP disclosed
WO-2007028456-A1 SUBSTITUTED PYRIDOCARBOXAMIDES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR 1 (PAI-1) BAYER HEALTHCARE AG (DE) 2007-03-15 WO disclosed