SCHEMBL4600535

SCHEMBL4600535

COC1(Br)C=CC(c2cccc(C(F)(F)F)c2)C=C1C=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.36
RCOR1 Q9UKL0 1/20 0.36
GUSB P08236 1/20 0.36
LMNA P02545 2/20 0.35
CYP2C19 P33261 1/20 0.35
TRPM5 Q9NZQ8 1/20 0.35
MAOB P27338 1/20 0.34
CACNA1F O60840 2/20 0.33
CACNA1D Q01668 2/20 0.33
CACNA1S Q13698 2/20 0.33
CACNA1C Q13936 2/20 0.33
POLB P06746 3/20 0.33
ALDH1A1 P00352 3/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HTR2C P28335 3/20 0.33
NQO2 P16083 1/20 0.32
MAPT P10636 3/20 0.32
KDM4E B2RXH2 1/20 0.32
DRD2 P14416 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5318529 0.69 KDM1A (0.43) KDM1ARCOR1HTR2CDRD2HTR2A
SCHEMBL4600218 0.64
SCHEMBL6984973 0.62 RIPK1 (0.32)
SCHEMBL11865252 0.61 GUSB (0.47) GUSBLMNACYP2C19TRPM5CACNA1F
SCHEMBL10601313 0.60 HTR2C (0.50) KDM1ARCOR1HTR2CDRD2HTR2A
SCHEMBL67201 0.60 FBP1 (0.56) LMNAMAOBPOLBALDH1A1L3MBTL1
SCHEMBL29425705 0.60 FBP1 (0.56) LMNAMAOBPOLBALDH1A1L3MBTL1
Acetaldehyde SCHEMBL28151033 0.59 NFE2L2 (0.54) LMNAMAOBPOLBALDH1A1L3MBTL1
SCHEMBL8702459 0.59 NFE2L2 (0.58) LMNAMAOBPOLBALDH1A1L3MBTL1
SCHEMBL9377104 0.58 HTR2C (0.44) KDM1ARCOR1LMNACYP2C19HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910292-A1 PIPERIDINE DERIVATIVE AS TACHYKININ RECEPTOR ANTAGONIST Takeda Pharmaceutical Company Limited (JP) 2008-04-16 EP disclosed
WO-2007015588-A1 PIPERIDINE DERIVATIVE AS TACHYKININ RECEPTOR ANTAGONIST TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-08 WO disclosed