SCHEMBL4600628

SCHEMBL4600628

C=CC(=O)Oc1c(OCCOC)cccc1Oc1ccc(N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.47
THRB P10828 4/20 0.36
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
THRA P10827 1/20 0.34
BTK Q06187 2/20 0.33
ITK Q08881 2/20 0.33
JAK2 O60674 1/20 0.33
LYN P07948 1/20 0.33
TEC P42680 1/20 0.33
TXK P42681 1/20 0.33
BMX P51813 1/20 0.33
JAK3 P52333 1/20 0.33
CD69 Q07108 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4600425 0.85 MAPT (0.46) EGFRGAAL3MBTL1LMNAMAPT
SCHEMBL4600130 0.83 EGFR (0.47) EGFRTHRBKDM4ELMNAMEN1
SCHEMBL4602781 0.81 EGFR (0.45) EGFRKDM4EMEN1KMT2ABTK
SCHEMBL4601601 0.79 EGFR (0.47) EGFRTHRBGAAKDM4ELMNA
SCHEMBL4602183 0.78 EGFR (0.47) EGFRTHRBGAAL3MBTL1MAPT
SCHEMBL4601033 0.77 EGFR (0.44) EGFRTHRBKDM4ETHRA
SCHEMBL4614803 0.75 EGFR (0.42) EGFRTHRBTHRAITK
SCHEMBL4601414 0.75 EGFR (0.44) EGFRL3MBTL1KDM4ELMNAITK
SCHEMBL4602178 0.75 EGFR (0.43) EGFRKDM4ELMNAMEN1KMT2A
SCHEMBL4602169 0.75 EGFR (0.41) EGFRKDM4EKMT2AITKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912645-A2 THERAPEUTIC AGENT FOR DIABETES Takeda Pharmaceutical Company Limited (JP) 2008-04-23 EP disclosed
WO-2007018314-A2 THERAPEUTIC AGENT FOR DIABETES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-15 WO disclosed