SCHEMBL4601033

SCHEMBL4601033

C=CC(=O)Oc1c(OCCOC)cccc1OCC1CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.44
PDE4B Q07343 4/20 0.43
PDE4A P27815 3/20 0.43
PDE4C Q08493 3/20 0.43
PDE4D Q08499 3/20 0.43
HTR2A P28223 1/20 0.38
GRM2 Q14416 1/20 0.38
RIPK1 Q13546 1/20 0.36
THRB P10828 2/20 0.35
THRA P10827 1/20 0.35
CNR2 P34972 2/20 0.35
FAAH O00519 1/20 0.35
CNR1 P21554 1/20 0.35
MRGPRX1 Q96LB2 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
KDR P35968 1/20 0.34
ACACB O00763 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4600070 0.94 EGFR (0.42) EGFRPDE4BPDE4APDE4CPDE4D
SCHEMBL4601672 0.84 SMN1; SMN2 (0.41) EGFRTHRB
SCHEMBL4602061 0.83 PDE4B (0.42) EGFRPDE4BPDE4APDE4CPDE4D
SCHEMBL4601601 0.81 EGFR (0.47) EGFRHTR2AGRM2THRBTHRA
SCHEMBL4600130 0.80 EGFR (0.47) EGFRHTR2AGRM2THRBTHRA
SCHEMBL4602183 0.80 EGFR (0.47) EGFRTHRB
SCHEMBL4631636 0.79 PDE4B (0.43) EGFRPDE4BPDE4APDE4CPDE4D
SCHEMBL4600628 0.77 EGFR (0.47) EGFRTHRBTHRAKDM4E
SCHEMBL4600843 0.76 RAB9A (0.50) EGFRKDM4E
SCHEMBL27368198 0.76 KCNK3 (0.42) EGFRTHRBTHRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912645-A2 THERAPEUTIC AGENT FOR DIABETES Takeda Pharmaceutical Company Limited (JP) 2008-04-23 EP disclosed
WO-2007018314-A2 THERAPEUTIC AGENT FOR DIABETES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-15 WO disclosed