SCHEMBL4603116

SCHEMBL4603116

C#CCOc1ccc(C(=O)NC2CC2)c(C)c1F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 4/20 0.40
HTR2A P28223 1/20 0.40
CNR1 P21554 3/20 0.39
CNR2 P34972 3/20 0.39
TAS1R3 Q7RTX0 6/20 0.39
TAS1R1 Q7RTX1 5/20 0.39
TAS1R2 Q8TE23 5/20 0.39
P2RX7 Q99572 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4603858 0.95 CNR1 (0.42) ALDH1A1POLBHPGDHTR2ACNR1
SCHEMBL4602882 0.95 CNR1 (0.44) ALDH1A1HPGDCNR1CNR2TAS1R3
SCHEMBL4603249 0.86 HTR2A (0.41) ALDH1A1POLBHPGDHTR2ACNR1
SCHEMBL4602587 0.82 HPGD (0.42) ALDH1A1POLBHPGDHTR2ACNR1
SCHEMBL4603506 0.82 HPGD (0.45) ALDH1A1HPGDHTR2ACNR1CNR2
SCHEMBL4604443 0.81 TAS1R3 (0.50) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL4604358 0.78 TAS1R3 (0.41) ALDH1A1POLBHPGDHTR2ACNR1
SCHEMBL4604804 0.77 HTR2A (0.35) ALDH1A1HTR2AP2RX7
SCHEMBL4604866 0.76 ALDH1A1 (0.51) ALDH1A1POLBHPGDCNR1CNR2
SCHEMBL4604028 0.76 ALDH1A1 (0.48) ALDH1A1POLBHPGDCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940780-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL CO., LTD. (JP) 2008-07-09 EP disclosed
WO-2007049728-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-03 WO disclosed