SCHEMBL4603249

SCHEMBL4603249

C#CCOc1ccc(C(=O)NC2CC2)c(CC)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.41
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 4/20 0.39
TAS1R3 Q7RTX0 2/20 0.37
TAS1R1 Q7RTX1 2/20 0.37
TAS1R2 Q8TE23 2/20 0.37
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
P2RX7 Q99572 1/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
PDE4B Q07343 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
SGMS2 Q8NHU3 1/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
HTR7 P34969 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4603506 0.96 HPGD (0.45) HTR2AALDH1A1HPGDCNR1CNR2
SCHEMBL4602587 0.96 HPGD (0.42) HTR2AALDH1A1POLBHPGDCNR1
SCHEMBL4604358 0.88 TAS1R3 (0.41) HTR2AALDH1A1POLBHPGDTAS1R3
SCHEMBL4603116 0.86 ALDH1A1 (0.42) HTR2AALDH1A1POLBHPGDTAS1R3
SCHEMBL4602808 0.84 HPGD (0.44) ALDH1A1HPGDCNR1CNR2
SCHEMBL4605222 0.84 HPGD (0.41) HTR2AALDH1A1HPGDCNR1CNR2
SCHEMBL4604638 0.83 ALDH1A1 (0.46) ALDH1A1HPGDCNR1CNR2
SCHEMBL4602882 0.82 CNR1 (0.44) ALDH1A1HPGDTAS1R3TAS1R1TAS1R2
SCHEMBL4603858 0.82 CNR1 (0.42) HTR2AALDH1A1POLBHPGDTAS1R3
SCHEMBL4603371 0.81 HPGD (0.42) HTR2AALDH1A1POLBHPGDCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940780-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL CO., LTD. (JP) 2008-07-09 EP disclosed
WO-2007049728-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-03 WO disclosed