SCHEMBL460502

SCHEMBL460502

CCn1c(-c2cncc3ccccc23)nc2c(F)c(F)ccc21

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 10/20 0.56
CYP11B1 P15538 8/20 0.40
NOS2 P35228 2/20 0.38
PTGER4 P35408 3/20 0.38
ERN1 O75460 1/20 0.37
HTR2C P28335 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
PRKCZ Q05513 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
RPS6KA5 O75582 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460601 0.85 CYP11B2 (0.67) CYP11B2CYP11B1ERN1PRKCZ
SCHEMBL17896589 0.80 CYP11B2 (0.51) CYP11B2CYP11B1HTR2CKDM4ERPS6KA5
SCHEMBL433566 0.79 RPS6KA5 (0.49) CYP11B2CYP11B1PTGER4HTR2CKDM4E
SCHEMBL10175445 0.72 CYP11B2 (1.00) CYP11B2CYP11B1ERN1PRKCZ
SCHEMBL17896650 0.70 PTGER4 (0.43) CYP11B2CYP11B1PTGER4KDM4EL3MBTL1
SCHEMBL17896768 0.70 CYP11B2 (0.69) CYP11B2CYP11B1NOS2ERN1NOS3
SCHEMBL461417 0.65 PDE10A (0.46) CYP11B2CYP11B1NOS2
SCHEMBL17883785 0.65 KDM4E (0.49) CYP11B2CYP11B1KDM4ERPS6KA5
SCHEMBL17896743 0.65 CYP11B2 (0.60) CYP11B2CYP11B1ERN1KDM4EMAPT
SCHEMBL11077028 0.65 NLRP3 (0.55) PTGER4KDM4EMAPTL3MBTL1RPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP claimed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO claimed