SCHEMBL4605834

SCHEMBL4605834

CC(O)C(Oc1cccc2[nH]c3ccccc3c12)N1CCN(C(=O)Cc2ccsc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
MAPT P10636 4/20 0.39
KDM4E B2RXH2 2/20 0.39
PKM P14618 1/20 0.39
ADRB3 P13945 7/20 0.38
ADRB2 P07550 7/20 0.38
ADRB1 P08588 6/20 0.38
HSD17B10 Q99714 3/20 0.38
DNM1 Q05193 1/20 0.37
POLB P06746 2/20 0.37
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607185 0.87 ADRB3 (0.46) CYP1A2CYP2C9CYP2C19MAPTKDM4E
SCHEMBL4608053 0.85 MAPT (0.50) MAPTADRB3ADRB2ADRB1HSD17B10
SCHEMBL4608603 0.84 ADRB3 (0.49) KDM4EADRB3ADRB2ADRB1ALDH1A1
SCHEMBL4606968 0.83 ADRB3 (0.42) MAPTADRB3ADRB2ADRB1HSD17B10
SCHEMBL4607632 0.83 MET (0.41) CYP1A2CYP2C9CYP2C19MAPTADRB3
SCHEMBL2991230 0.81 ADRB3 (0.58) ADRB3ADRB2ADRB1DNM1
SCHEMBL4608607 0.79 ALDH1A1 (0.44) CYP2C9CYP2C19PKMADRB3ADRB2
SCHEMBL4605132 0.77 ADRB3 (0.46) MAPTKDM4EADRB3ADRB2ADRB1
SCHEMBL4607629 0.77 KDM4E (0.52) CYP1A2CYP2C9CYP2C19MAPTKDM4E
SCHEMBL4607514 0.76 ADRB3 (0.49) KDM4EADRB3ADRB2ADRB1DNM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP disclosed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO disclosed