SCHEMBL4608607

SCHEMBL4608607

CC(O)C(Oc1cccc2[nH]c3ccccc3c12)N1CCN(C(=O)c2cccs2)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
LMNA P02545 2/20 0.44
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KCNA5 P22460 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 1/20 0.40
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PKM P14618 1/20 0.39
HTT P42858 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607733 0.88 POLB (0.40) ALDH1A1LMNASMN1; SMN2HSD17B10HTT
SCHEMBL4607629 0.82 KDM4E (0.52) ALDH1A1LMNACYP2C9CYP2C19SMN1; SMN2
SCHEMBL4606968 0.80 ADRB3 (0.42) LMNAHSD17B10ADRB2ADRB1ADRB3
SCHEMBL4605749 0.80 TLR9 (0.49) ALDH1A1LMNACYP2C19SMN1; SMN2GAA
SCHEMBL4608590 0.80 RAB9A (0.46) ALDH1A1LMNACYP2D6CYP2C9CYP2C19
SCHEMBL2994138 0.79 ADRB2 (0.60) KCNA5ADRB2ADRB1ADRB3
SCHEMBL4605834 0.79 CYP1A2 (0.44) ALDH1A1CYP2D6CYP2C9CYP2C19HSD17B10
SCHEMBL4607479 0.79 PTK2 (0.45) ADRB2ADRB1ADRB3
SCHEMBL4605132 0.78 ADRB3 (0.46) GAAADRB2ADRB1ADRB3
SCHEMBL4608251 0.78 MITF (0.43) ALDH1A1L3MBTL1PKMADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed