SCHEMBL460599

SCHEMBL460599

Fn1cnc2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.54
HTT P42858 3/20 0.52
CYP11B1 P15538 3/20 0.47
CYP11B2 P19099 3/20 0.47
POLB P06746 1/20 0.47
TNF P01375 1/20 0.47
FGFR1 P11362 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 2/20 0.44
MEN1 O00255 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
STAT6 P42226 1/20 0.44
ALDH3A1 P30838 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4388741 0.76 TDP1 (0.54) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL7196401 0.75 TDP1 (0.58) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL11706281 0.74 TDP1 (0.52) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL2489876 0.73 TDP1 (0.56) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL8668369 0.71 TDP1 (0.54) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL145442 0.71 TDP1 (0.54) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL5399 0.71 TDP1 (0.59) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL278161 0.71 TDP1 (0.54) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL277760 0.71 TDP1 (0.54) TDP1HTTCYP11B1CYP11B2POLB
SCHEMBL9062626 0.71 TDP1 (0.54) TDP1HTTCYP11B1CYP11B2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108640878-A A kind of BenzoiminazoleflouriAnd class compound and its preparation method and application 上海泰坦科技股份有限公司 2018-10-12 CN claimed
US-20260125376-A1 IRREVERSIBLE INACTIVATORS TARGETING ARAF/MEK COMPLEXES GERO THOMAS (US) 2026-05-07 US disclosed
CN-120172974-A 1-Fluorobenzimidazole pyridine derivative and preparation method and application thereof 淮阴师范学院 2025-06-20 CN disclosed
CN-120172974-A 1-Fluorobenzimidazole pyridine derivative and preparation method and application thereof 淮阴师范学院 2025-06-20 CN disclosed
US-20220403229-A1 ELECTRONIC CONTROL OF TRANSMITTANCE OF VISIBLE AND NEAR-INFRARED RADIATION KEBOTIX, INC. (US) 2022-12-22 US disclosed
CN-115350179-A Application of fluorobenzimidazole thiosemicarbazide compound in antitumor drugs 青岛科技大学 2022-11-18 CN disclosed
CN-109071508-A Benzimidazole bis-indole compound as novel divalent IAP antagonist 南京明德新药研发股份有限公司 2018-12-21 CN disclosed
CN-107312056-A The synthetic method of 2 (the pregnane base of 3 ' hydroxyl 17 ') 5 fluorobenzimidazoles 广西师范学院 2017-11-03 CN disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
CN-105142623-A Methods and compositions for improving cognitive function AGENEBIO INC 2015-12-09 CN disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed
EP-2298770-A1 Heterocyclic compounds as TrkA modulators ChemBridge Corporation (US) 2011-03-23 EP disclosed
US-20090105400-A1 Imidazolium side chains for example; for example polymers based on 1-methyl-3-(2H,9H,9H-perfluoro-3,6-dioxa-5-methyl-8-nonenyl)-imidazolium trifluoromethanesulfonate; polymer electrolytes for fuel cell, secondary battery, capacitor, dye-sensitized solar cell and electrochromic device DAIKIN INDUSTRIES, LTD. (JP) 2009-04-23 US disclosed
US-20090069343-A1 Combination Histamine H1R and H4R Antagonist Therapy for Treating Pruritus DUNFORD PAUL J 2009-03-12 US disclosed
US-20080207635-A1 Heterocyclic compounds useful in the treatment of neoplastic diseases, inflammatory disorders and immunomodulatory disorders CHEMBRIDGE CORPORATION 2008-08-28 US disclosed
EP-1960382-A1 HETEROCYCLIC COMPOUNDS AS TYROSINE KINASE MODULATORS ChemBridge Research Laboratories, Inc. (US) 2008-08-27 EP disclosed
WO-2007056155-A1 HETEROCYCLIC COMPOUNDS AS TYROSINE KINASE MODULATORS CHEMBRIDGE RESEARCH LABORATORIES, INC. (US) 2007-05-18 WO disclosed
CN-1784387-A Novel benzimidazole derivatives ASTRAZENECA AB (SE) 2006-06-07 CN disclosed
US-5118506-A Mixing with baits in solid or liquid forms which acts as a poison to kill fire ants by ingestion or by respiratory contact; nontoxic to human and animal Casella, Peter F. (US) 1992-06-02 US disclosed
US-4891222-A AQUEOUS EMULSION, NONIONIC AND ANIONIC SURFACTANTS TFA PRODUCTS, INC 1990-01-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260125376-A1 IRREVERSIBLE INACTIVATORS TARGETING ARAF/MEK COMPLEXES ARAF, BRAF, RAF1 TDP1 2570/4885HTT 3759/4885CYP11B1 3242/4885
US-20080207635-A1 Heterocyclic compounds useful in the treatment of neoplastic diseases, inflammatory disorders and immunomodulatory disorders LCK, MALT1, MYD88 TDP1 1277/4885HTT 2486/4885CYP11B1 913/4885
US-20090069343-A1 Combination Histamine H1R and H4R Antagonist Therapy for Treating Pruritus HRH4, HRH2, HRH3 TDP1 3094/4885HTT 563/4885CYP11B1 3706/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.