SCHEMBL4608279

SCHEMBL4608279

Oc1ccnc(SCCCN2CCN(c3cccc(C(F)(F)F)c3)CC2)n1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.53
DRD3 P35462 7/20 0.53
ADRA1A P35348 4/20 0.53
HRH4 Q9H3N8 1/20 0.53
SIGMAR1 Q99720 2/20 0.52
HTR7 P34969 4/20 0.52
DRD5 P21918 1/20 0.50
HTR1A P08908 1/20 0.49
HTR2A P28223 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674560 0.85 DRD2 (0.62) DRD2DRD3ADRA1AHRH4SIGMAR1
SCHEMBL4610058 0.83 DHFR (0.46) DRD2DRD3ADRA1AHRH4SIGMAR1
SCHEMBL4610053 0.83 DHFR (0.46) DRD2DRD3ADRA1AHRH4SIGMAR1
Hydrochloric Acid SCHEMBL4609800 0.83 DHFR (0.45) DRD2DRD3ADRA1AHRH4SIGMAR1
Hydrochloric Acid SCHEMBL7070981 0.83 DHFR (0.45) DRD2DRD3ADRA1AHRH4SIGMAR1
Hydrochloric Acid SCHEMBL4609803 0.83 DHFR (0.45) DRD2DRD3ADRA1AHRH4SIGMAR1
Hydrochloric Acid SCHEMBL7070972 0.83 DHFR (0.45) DRD2DRD3ADRA1AHRH4SIGMAR1
SCHEMBL4608233 0.82 KCNH2 (0.40) DRD2DRD3HTR7DRD5HTR1A
SCHEMBL2437211 0.81 DRD2 (0.49) DRD2DRD3HTR1AHTR2A
SCHEMBL7047571 0.80 DRD2 (0.64) DRD2DRD3ADRA1AHRH4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1272187-B1 DOPAMINE-D3 RECEPTOR LIGANDS FOR THE TREATMENT OF ADDICTION ABBOTT GMBH & CO KG (DE) 2008-07-30 EP claimed
EP-1272187-B1 DOPAMINE-D3 RECEPTOR LIGANDS FOR THE TREATMENT OF ADDICTION ABBOTT GMBH & CO KG (DE) 2008-07-30 EP disclosed