SCHEMBL4610053

SCHEMBL4610053

Oc1ccnc(SC/C=C/CN2CCN(c3cccc(C(F)(F)F)c3)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.46
KDM4E B2RXH2 4/20 0.45
POLB P06746 2/20 0.45
PHGDH O43175 2/20 0.44
DRD2 P14416 4/20 0.44
DRD3 P35462 4/20 0.44
ADRA1A P35348 3/20 0.44
HRH4 Q9H3N8 1/20 0.44
HTR1A P08908 1/20 0.44
MAPT P10636 4/20 0.43
LMNA P02545 3/20 0.43
GAA P10253 2/20 0.43
SIGMAR1 Q99720 1/20 0.43
XBP1 P17861 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
HSP90AA1 P07900 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4610058 1.00 DHFR (0.46) DHFRKDM4EPOLBPHGDHDRD2
Hydrochloric Acid SCHEMBL7070981 0.99 DHFR (0.45) DHFRKDM4EPOLBPHGDHDRD2
Hydrochloric Acid SCHEMBL4609800 0.99 DHFR (0.45) DHFRKDM4EPOLBPHGDHDRD2
Hydrochloric Acid SCHEMBL7070972 0.99 DHFR (0.45) DHFRKDM4EPOLBPHGDHDRD2
Hydrochloric Acid SCHEMBL4609803 0.99 DHFR (0.45) DHFRKDM4EPOLBPHGDHDRD2
SCHEMBL4608279 0.83 DRD2 (0.53) DRD2DRD3ADRA1AHRH4HTR1A
SCHEMBL8560485 0.74 SIGMAR1 (0.56) DHFRKDM4EPOLBHTR1AMAPT
SCHEMBL8560489 0.74 SIGMAR1 (0.56) DHFRKDM4EPOLBHTR1AMAPT
SCHEMBL8577276 0.70 SIGMAR1 (0.60) KDM4EPOLBHTR1AMAPTLMNA
SCHEMBL1733940 0.70 SIGMAR1 (0.60) KDM4EPOLBHTR1AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1272187-B1 DOPAMINE-D3 RECEPTOR LIGANDS FOR THE TREATMENT OF ADDICTION ABBOTT GMBH & CO KG (DE) 2008-07-30 EP claimed