SCHEMBL4608922

SCHEMBL4608922

CC1=C(C(=O)O)C(CC(C)C)(c2ccccc2[N+](=O)[O-])C(C(=O)O)=C(C)N1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.38
POLB P06746 2/20 0.38
TDP1 Q9NUW8 2/20 0.37
TSHR P16473 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
FBP1 P09467 1/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 4/20 0.35
CYP2C9 P11712 1/20 0.35
CYP3A4 P08684 1/20 0.34
ABCC4 O15439 1/20 0.34
CACNA1F O60840 1/20 0.34
NR1I2 O75469 1/20 0.34
ABCB11 O95342 1/20 0.34
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
ABCB1 P08183 1/20 0.34
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755372 0.76 TSHR (0.39) POLBTDP1TSHRL3MBTL1FBP1
SCHEMBL7274724 0.75 CACNA1B (0.38) TSHRFBP1LMNA
SCHEMBL7382729 0.74 TSHR (0.37) POLBTDP1TSHRL3MBTL1ALDH1A1
SCHEMBL8896632 0.70 TSHR (0.42) POLBTDP1TSHRL3MBTL1ALDH1A1
SCHEMBL4880017 0.68 TSHR (0.38) POLBTDP1TSHRL3MBTL1ALDH1A1
SCHEMBL3396115 0.67 GPR35 (0.41) CYP2C19POLBTDP1TSHRL3MBTL1
SCHEMBL7351539 0.66 MAPT (0.37) POLBTDP1TSHRL3MBTL1ALDH1A1
SCHEMBL4880853 0.65 ABCC4 (0.47) CYP2C19POLBTDP1TSHRALDH1A1
SCHEMBL27819930 0.64 POLB (0.52) CYP2C19POLBTDP1TSHRL3MBTL1
SCHEMBL2944564 0.63 HSD17B10 (0.39) CYP2C19POLBTDP1TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532110-B1 INDUSTRIAL PROCESS FOR THE SYNTHESIS OF ISOBUTYL METHYL 1,4-DIHYDRO-2,6-DIMETHYL-4-(2-NITROPHENYL)-3,5-PYRIDINE DICARBOXYLATE (NISOLDIPINE) ERREGIERRE SPA (IT) 2008-07-23 EP claimed