SCHEMBL4880853

SCHEMBL4880853

CC1=C(C(=O)O)C(c2ccccc2[N+](=O)[O-])C(C(=O)O)=C(C)N1CCC(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC4 O15439 2/20 0.47
CACNA1F O60840 2/20 0.47
ABCB11 O95342 2/20 0.47
LMNA P02545 2/20 0.47
CYP1A2 P05177 2/20 0.47
ADORA3 P0DMS8 2/20 0.47
ADORA2A P29274 2/20 0.47
ADORA1 P30542 2/20 0.47
OPRM1 P35372 2/20 0.47
SCN1A P35498 2/20 0.47
HTR2B P41595 2/20 0.47
CACNA1D Q01668 2/20 0.47
KCNH2 Q12809 2/20 0.47
CACNA1S Q13698 2/20 0.47
CACNA1C Q13936 2/20 0.47
SCN5A Q14524 2/20 0.47
SCN2A Q99250 2/20 0.47
SCN3A Q9NY46 2/20 0.47
NR1I2 O75469 1/20 0.47
NR3C1 P04150 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5414545 0.90 ALDH1A1 (0.45) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL5414539 0.90 ALDH1A1 (0.45) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL28318011 0.88 ADORA3 (0.49) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL11007311 0.83 ALDH1A1 (0.43) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL10516391 0.83 ALDH1A1 (0.51) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL10516412 0.83 ALDH1A1 (0.51) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL28770058 0.82 ALDH1A1 (0.48) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL10553898 0.80 PYGL (0.52) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL11009925 0.80 ALDH1A1 (0.45) ABCC4CACNA1FABCB11LMNACYP1A2
SCHEMBL4880010 0.80 CACNA1C (0.46) ABCC4CACNA1FABCB11LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080095841-A1 Pharmaceutical Composition, Method for Producing the Same, and Method for Stabilizing Dihydropyridine Compound in the Pharmaceutical Composition EISAI R&D MANAGEMENT CO., LTD. (JP) 2008-04-24 US disclosed
EP-1813274-A1 MEDICINAL COMPOSITION, PROCESS FOR PRODUCING THE SAME, AND METHOD OF STABILIZING DIHYDROPYRIDINE COMPOUND IN MEDICINAL COMPOSITION Eisai R&D Management Co., Ltd. (JP) 2007-08-01 EP disclosed