SCHEMBL3396115

SCHEMBL3396115

CCN1C(C)=C(C(=O)O)C(CC)(c2cccc([N+](=O)[O-])c2O)C(C(=O)O)=C1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.41
TDP1 Q9NUW8 3/20 0.40
TSHR P16473 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
MAPT P10636 5/20 0.36
ALDH1A1 P00352 5/20 0.36
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
FBP1 P09467 1/20 0.36
ERN1 O75460 1/20 0.35
CXCR1 P25024 1/20 0.35
CXCR2 P25025 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
POLB P06746 2/20 0.34
GLA P06280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755372 0.91 TSHR (0.39) TDP1TSHRL3MBTL1MAPTALDH1A1
SCHEMBL3392997 0.76 TDP1 (0.40) TDP1L3MBTL1MAPTALDH1A1MEN1
SCHEMBL4757355 0.75 PYGM (0.39) CRHBPCRHR2ALDH1A1CYP2C19LMNA
SCHEMBL4755316 0.75 HCAR2 (0.36) TSHRALDH1A1MEN1KMT2ARECQL
SCHEMBL4758299 0.73 LMNA (0.42) TDP1TSHRALDH1A1MEN1KMT2A
SCHEMBL11390110 0.72 TDP1 (0.37) TDP1L3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL9826311 0.69 CYSLTR2 (0.40) CRHBPCRHR2MAPTALDH1A1KMT2A
SCHEMBL6385093 0.69 TPMT (0.35) MAPTALDH1A1MEN1KMT2A
SCHEMBL7429615 0.68 TDP1 (0.37) TDP1TSHRL3MBTL1MAPTALDH1A1
SCHEMBL4880017 0.68 TSHR (0.38) TDP1TSHRL3MBTL1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229167-A1 MINERALOCORTICOID RECEPTOR MODULATORS Merck Sharp & Dohme Corp. (US) 2010-09-22 EP claimed
WO-2009078934-A1 MINERALOCORTICOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2009-06-25 WO claimed