SCHEMBL4617893

SCHEMBL4617893

O=S(=O)(Cl)c1cc(S(=O)(=O)c2ccccc2F)ccc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.48
HTR2C P28335 3/20 0.46
HTR2B P41595 1/20 0.46
SLC22A12 Q96S37 3/20 0.43
ABCC9 O60706 1/20 0.42
ABCC8 Q09428 1/20 0.42
KCNJ11 Q14654 1/20 0.42
KCNJ8 Q15842 1/20 0.42
HTR2A P28223 6/20 0.42
CNR1 P21554 4/20 0.41
KCNH2 Q12809 2/20 0.41
WNT3 P56703 1/20 0.41
SFRP1 Q8N474 1/20 0.41
CNR2 P34972 3/20 0.41
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4615993 0.84 SFRP1 (0.55) HSD11B1WNT3SFRP1
SCHEMBL4616786 0.81 HSD11B1 (0.49) HSD11B1HTR2CHTR2BSLC22A12ABCC9
SCHEMBL4616832 0.81 HSD11B1 (0.45) HSD11B1HTR2CHTR2BABCC9ABCC8
SCHEMBL4617928 0.78 KMT2A (0.54) HSD11B1HTR2CHTR2BABCC9ABCC8
SCHEMBL4617061 0.77 HSD11B1 (0.54) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL65955 0.74 MEN1 (0.56) HSD11B1SLC22A12CYP2C9
SCHEMBL29500393 0.74 MEN1 (0.56) HSD11B1SLC22A12CYP2C9
SCHEMBL6101134 0.74 SFRP1 (0.60) WNT3SFRP1
SCHEMBL27713242 0.74 SLC22A12 (0.34) HSD11B1SLC22A12WNT3SFRP1
SCHEMBL4616747 0.73 PKM (0.53) HSD11B1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof SFRP1, SOS1, FZD7 HSD11B1 205/4885HTR2C 3668/4885HTR2B 3802/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.