SCHEMBL4621546

SCHEMBL4621546

COc1ccc(C(=O)S(=O)(=O)NCC(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.52
CA1 P00915 6/20 0.49
CA2 P00918 6/20 0.49
TSHR P16473 1/20 0.48
PARP1 P09874 1/20 0.47
PARP10 Q53GL7 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
PARP4 Q9UKK3 1/20 0.47
PDE4B Q07343 1/20 0.46
CES2 O00748 2/20 0.46
CES1 P23141 2/20 0.46
HSD11B1 P28845 1/20 0.46
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
PLK1 P53350 1/20 0.45
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4185509 0.82 PARP1 (0.53) MAPTPARP1CES2CES1HSD11B1
SCHEMBL4163523 0.80 MMP12 (0.50) MAPTTSHRPARP1CES1KDM4E
SCHEMBL7674553 0.79 HSD11B1 (0.57) MAPTCA1CA2TSHRPDE4B
SCHEMBL4173740 0.78 MEP1B (0.67) MAPTCA1CA2TSHRHTT
SCHEMBL1732559 0.74 HTT (0.72) MAPTCA2TSHRHTTCA12
SCHEMBL4622173 0.74 CA1 (0.47) CA1CA2PARP1PARP10PARP2
SCHEMBL4621268 0.74 CA1 (0.47) CA1CA2PARP1PARP10PARP2
SCHEMBL4620575 0.74 CA1 (0.47) CA1CA2PARP1PARP10PARP2
SCHEMBL4621422 0.74 CA2 (0.46) CA1CA2PARP1PARP10PARP2
SCHEMBL4620569 0.74 CA2 (0.46) CA1CA2PARP1PARP10PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1884230-A1 PARAKERATOSIS INHIBITOR, PORE-SHRINKING AGENT OR AGENT FOR PREVENTING/AMELIORATING ROUGH SKIN AND EXTERNAL COMPOSITION FOR SKIN Shiseido Company, Limited (JP) 2008-02-06 EP disclosed