SCHEMBL4627490

SCHEMBL4627490

COc1cccc(OC)c1-c1ccc2cc(CC(C)(NC(=O)[C@@H]3CCCN3S(=O)(=O)c3ccccc3)C(=O)O)ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 14/20 0.49
ITGB7 P26010 12/20 0.49
TDP1 Q9NUW8 1/20 0.49
ITGB1 P05556 5/20 0.49
HCRTR1 O43613 2/20 0.46
HCRTR2 O43614 2/20 0.46
RAB9A P51151 1/20 0.46
KCNQ1 P51787 2/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3314005 0.83 ITGA4 (0.65) ITGA4ITGB7ITGB1
SCHEMBL3317078 0.82 ITGA4 (0.57) ITGA4ITGB7ITGB1
SCHEMBL5175652 0.79 L3MBTL1 (0.42) ITGA4ITGB7ITGB1HCRTR1HCRTR2
SCHEMBL6141659 0.78 ITGA4 (0.54) ITGA4ITGB7ITGB1
SCHEMBL4625291 0.77 ITGB1 (0.39) ITGA4ITGB7TDP1ITGB1LMNA
SCHEMBL3859283 0.76 ITGA4 (0.75) ITGA4ITGB7ITGB1
SCHEMBL4624059 0.73 ITGA4 (0.50) ITGA4ITGB7TDP1ITGB1LMNA
SCHEMBL13570517 0.69 FKBP1A (0.69) TDP1HCRTR1HCRTR2RAB9A
SCHEMBL13570871 0.69 TDP1 (0.69) TDP1RAB9ASMN1; SMN2
SCHEMBL6140371 0.69 ITGA4 (0.53) ITGA4ITGB7ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP claimed