SCHEMBL462885

SCHEMBL462885

CC1=NNC(c2cccc(F)c2)C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.57
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
IDO1 P14902 1/20 0.40
MAOB P27338 2/20 0.40
MAOA P21397 1/20 0.40
TAAR1 Q96RJ0 1/20 0.38
NOS3 P29474 1/20 0.38
RIPK1 Q13546 1/20 0.37
ACHE P22303 1/20 0.37
KDM1A O60341 1/20 0.37
RCOR1 Q9UKL0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23146476 0.83 CA1 (0.38) CA1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL9037008 0.79 MAOA (0.44) CA1SMN1; SMN2KDM4EMAPTMAOB
SCHEMBL16500516 0.78 CA1 (0.57) CA1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL1660314 0.72 MAOA (0.61) CA1KDM4EMAPTMAOBMAOA
SCHEMBL13330945 0.71 ALDH1A1 (0.37) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL9378182 0.70 CA1 (0.46) CA1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL21523818 0.69 KDM4E (0.47) CA1KDM4EL3MBTL1HTR2AHTR2C
SCHEMBL172227 0.69 HTR2A (0.44) CA1IDO1TAAR1ACHEKDM1A
SCHEMBL21523837 0.68 CHRNB2 (0.48) CA1ALDH1A1TAAR1KDM1ARCOR1
SCHEMBL21723161 0.66 HTR2A (0.41) CA1KDM4EALDH1A1IDO1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012034095-A1 COMPOUNDS AND COMPOSITIONS AS TRK INHIBITORS IRM LLC (BM) 2012-03-15 WO disclosed
WO-2012034095-A1 COMPOUNDS AND COMPOSITIONS AS TRK INHIBITORS IRM LLC (BM) 2012-03-15 WO disclosed