SCHEMBL4629210

SCHEMBL4629210

COc1cc(Br)c(C)c(CC2(C3(Cc4c(C)cccc4Br)NCCN3)NCCN2)c1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ADORA2A P29274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630337 0.76 SLC6A2 (0.35) KDM4EALDH1A1
SCHEMBL4629208 0.71 HTR1D (0.56)
SCHEMBL4630003 0.64 P2RX7 (0.36)
SCHEMBL957652 0.62 CYP3A4 (0.40) ALDH1A1
SCHEMBL4630018 0.61 KMT2A (0.39) KDM4EALDH1A1
SCHEMBL4629824 0.59 TAAR1 (0.35)
SCHEMBL4297601 0.59 ALDH1A1 (0.56) ALDH1A1
SCHEMBL954687 0.58 HTR1B (0.52) KDM4E
SCHEMBL30550473 0.58 ALDH1A1 (0.48) ALDH1A1
SCHEMBL560310 0.57 IDO1 (0.33) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP claimed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO claimed
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed