SCHEMBL463041

SCHEMBL463041

COCCc1nc(-c2cc(F)cc(F)c2)[nH]c(=O)c1C(=O)C1C(=O)C2CCC(C2)C1=O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TNKS O95271 6/20 0.33
TNKS2 Q9H2K2 6/20 0.33
PARP1 P09874 5/20 0.33
CTSS P25774 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
KCNH2 Q12809 2/20 0.31
SMPD3 Q9NY59 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL454917 0.80 TNKS (0.41) TNKSTNKS2PARP1GRIN1GRIN2B
SCHEMBL9903971 0.67 CYP1A2 (0.40) GRIN1GRIN2B
SCHEMBL3234904 0.61 IRAK4 (0.31)
SCHEMBL13291364 0.61 HSD11B1 (0.32)
SCHEMBL454863 0.61 WNT3A (0.39) TNKS2
SCHEMBL13291842 0.61 TRPV1 (0.36) KCNH2
SCHEMBL13291801 0.60 TRPV1 (0.32)
SCHEMBL13291798 0.60 TRPV1 (0.32)
SCHEMBL30177122 0.59 DRD2 (0.32) KCNH2
SCHEMBL13383746 0.58 TRPV1 (0.32) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2475654-A1 HERBICIDAL PYRIMIDONE DERIVATIVES E. I. du Pont de Nemours and Company (US) 2012-07-18 EP disclosed
WO-2012033548-A2 HERBICIDAL BIS-NITROGEN-CONTAINING OXO AND SULFONO HETEROCYCLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-03-15 WO disclosed
WO-2011031658-A1 HERBICIDAL PYRIMIDONE DERIVATIVES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-03-17 WO disclosed