SCHEMBL4631483

SCHEMBL4631483

[CH2]Oc1cc(CC)cnc1Cl

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.34
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22641245 0.83 PTGS2 (0.48) PTGS2TDP1L3MBTL1PDE4APDE4B
SCHEMBL4881459 0.79 CRHR1 (0.33) PTGS2
SCHEMBL6603590 0.77 MAPT (0.38) NPC1RAB9A
SCHEMBL2853131 0.75 ALDH1A1 (0.32) TDP1
SCHEMBL8272903 0.74 ALDH1A1 (0.44) TDP1L3MBTL1POLB
SCHEMBL22978573 0.73 ALDH1A1 (0.37) TDP1PDE4APDE4DNPC1POLB
SCHEMBL6607673 0.73 CRHR1 (0.35)
SCHEMBL2597202 0.72 NOS3 (0.35)
SCHEMBL2851798 0.72 PDE4A (0.36) L3MBTL1PDE4APDE4BPDE4CPDE4D
SCHEMBL2853192 0.71 XPO1 (0.35) L3MBTL1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924558-A1 AN ANTIMALARIAL BAYLIS-HILLMAN ADDUCTS AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-05-28 EP disclosed
WO-2007032016-A1 AN ANTIMALARIAL BAYLIS-HILLMAN ADDUCTS AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2007-03-22 WO disclosed