SCHEMBL4631973

SCHEMBL4631973

CN(Cc1ccc(C#N)cc1)CC(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.46
NSD2 O96028 1/20 0.46
POLB P06746 1/20 0.44
LOXL2 Q9Y4K0 2/20 0.43
PYCR1 P32322 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
CYP19A1 P11511 1/20 0.39
ACHE P22303 2/20 0.38
MAOB P27338 2/20 0.38
IDO1 P14902 1/20 0.38
KIF11 P52732 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
LSS P48449 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
MLYCD O95822 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23015092 0.79 NSD2 (0.63) CYP2A6NSD2POLBLOXL2PYCR1
SCHEMBL12749574 0.78 PYCR1 (0.52) CYP2A6PYCR1IDO1HRH3
SCHEMBL23374744 0.78 CYP2A6 (0.57) CYP2A6NSD2POLBLOXL2SIGMAR1
SCHEMBL4632355 0.77 PYCR1 (0.41) LOXL2PYCR1MAOBHRH3
SCHEMBL21962259 0.77 PYCR1 (0.53) PYCR1MAOBLSS
SCHEMBL1472497 0.77 NR1I2 (0.42) PYCR1MAOBKIF11HRH3
SCHEMBL7039840 0.77 SIGMAR1 (0.57) CYP2A6PYCR1SIGMAR1TMEM97CRHBP
SCHEMBL1009445 0.77 PYCR1 (0.38) PYCR1SIGMAR1MAOBHRH3
SCHEMBL23032284 0.76 ALDH1A1 (0.52) PYCR1SIGMAR1MAOB
SCHEMBL156261 0.75 CYP2A6 (0.58) CYP2A6NSD2POLBLOXL2CRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924561-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS Eli Lilly & Company (US) 2008-05-28 EP disclosed
WO-2007028083-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2007-03-08 WO disclosed