SCHEMBL4633263

SCHEMBL4633263

O=C(O)c1scc(Nc2ccc(Br)cc2[N+](=O)[O-])c1OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 5/20 0.44
CTSL P07711 5/20 0.44
MAPT P10636 3/20 0.42
AKR1C3 P42330 2/20 0.42
AKR1C2 P52895 2/20 0.42
HCAR3 P49019 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP19A1 P11511 1/20 0.39
PKM P14618 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MYC P01106 1/20 0.38
MAX P61244 1/20 0.38
SENP5 Q96HI0 1/20 0.38
SENP2 Q9HC62 1/20 0.38
SENP1 Q9P0U3 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
AKR1B10 O60218 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4407305 0.82 CTSV (0.42) CTSVCTSLMAPTAKR1C3AKR1C2
SCHEMBL3607732 0.80 CTSV (0.48) CTSVCTSLMAPTAKR1C3AKR1C2
SCHEMBL3607727 0.80 CTSV (0.48) CTSVCTSLMAPTAKR1C3AKR1C2
SCHEMBL4633259 0.75 CTSV (0.43) CTSVCTSLMAPTCYP19A1MYC
SCHEMBL3255304 0.74 CTSV (0.44) CTSVCTSLMAPTAKR1C3AKR1C2
SCHEMBL29197789 0.73 PIN1 (0.46) CTSVCTSLMAPTSMN1; SMN2CYP19A1
SCHEMBL22711369 0.72 THRA (0.51) MAPTALDH1A1SMN1; SMN2L3MBTL1KMT2A
SCHEMBL6019985 0.71 ABCB1 (0.42) CTSVCTSLMAPTCYP19A1PKM
SCHEMBL8391099 0.70 AKR1C3 (0.71) CTSVCTSLMAPTAKR1C3AKR1C2
SCHEMBL31473699 0.70 POLB (0.57) CTSVCTSLMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924572-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SmithKline Beecham Corporation (US) 2008-05-28 EP disclosed
WO-2007030366-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed