SCHEMBL4635153

SCHEMBL4635153

C=C(O)CN(CC(=C)O)c1ccc(C)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.48
TSHR P16473 2/20 0.41
ALDH1A1 P00352 1/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
CNR2 P34972 4/20 0.36
ACHE P22303 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948375 0.85 CNR1 (0.41) CYP2C19TSHRALDH1A1KEAP1NFE2L2
SCHEMBL9974573 0.78 KEAP1 (0.56) CYP2C19ALDH1A1KEAP1NFE2L2CNR2
SCHEMBL145821 0.77 CYP2C19 (0.50) CYP2C19TSHRALDH1A1KEAP1NFE2L2
SCHEMBL33921 0.73 CYP2C19 (0.47) CYP2C19TSHRALDH1A1KEAP1NFE2L2
SCHEMBL17689350 0.71 ALDH1A1 (0.46) CYP2C19TSHRALDH1A1CNR2TDP1
SCHEMBL3348811 0.71 KEAP1 (0.49) CYP2C19TSHRKEAP1NFE2L2CNR2
SCHEMBL2805280 0.71 KMT2A (0.50) CYP2C19TSHRALDH1A1KEAP1NFE2L2
SCHEMBL7108072 0.70 ALDH1A1 (0.46) CYP2C19TSHRALDH1A1KEAP1NFE2L2
SCHEMBL516400 0.70 CYP2C19 (0.48) CYP2C19TSHRALDH1A1CNR2ACHE
Bicarbonate SCHEMBL11138673 0.70 CNR2 (0.56) CYP2C19TSHRALDH1A1CNR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9512298-B2 Specific mixtures of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS DEUTSCHLAND GMBH (DE) 2016-12-06 US disclosed
US-9512298-B2 Specific mixtures of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS DEUTSCHLAND GMBH (DE) 2016-12-06 US disclosed
US-9512298-B2 Specific mixtures of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS DEUTSCHLAND GMBH (DE) 2016-12-06 US disclosed
US-20130116395-A1 Specific mixtrues of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS Deutschland (DE) 2013-05-09 US disclosed
US-20130116395-A1 Specific mixtrues of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS Deutschland (DE) 2013-05-09 US disclosed
US-20130116395-A1 Specific mixtrues of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS Deutschland (DE) 2013-05-09 US disclosed
EP-1650184-B1 Mixtures of N,N-Bis-(2-hydroxyalkyl)-4-toluidin, their preparation and use SALTIGO GMBH (DE) 2008-01-23 EP disclosed
EP-1650184-B1 Mixtures of N,N-Bis-(2-hydroxyalkyl)-4-toluidin, their preparation and use SALTIGO GMBH (DE) 2008-01-23 EP disclosed
EP-1650184-A1 Mixtures of N,N-Bis-(2-hydroxyalkyl)-4-toluidin, their preparation and use Lanxess Deutschland GmbH (DE) 2006-04-26 EP disclosed
EP-1650184-A1 Mixtures of N,N-Bis-(2-hydroxyalkyl)-4-toluidin, their preparation and use Lanxess Deutschland GmbH (DE) 2006-04-26 EP disclosed
EP-1650184-A1 Mixtures of N,N-Bis-(2-hydroxyalkyl)-4-toluidin, their preparation and use Lanxess Deutschland GmbH (DE) 2006-04-26 EP disclosed
US-20060052555-A1 Specific mixtures of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS DEUTSCHLAND GMBH 2006-03-09 US disclosed
US-20060052555-A1 Specific mixtures of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS DEUTSCHLAND GMBH 2006-03-09 US disclosed
US-20060052555-A1 Specific mixtures of N,N-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS DEUTSCHLAND GMBH 2006-03-09 US disclosed
CN-1743364-A Specific mixtures of n,n-bis(2-hydroxyalkyl)-4-toluidine derivatives, their preparation and a method of using such specific mixtures LANXESS DEUTSCHLAND GMBH (DE) 2006-03-08 CN disclosed