SCHEMBL4637822

SCHEMBL4637822

O=C(C#Cc1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
ADORA3 P0DMS8 2/20 0.41
PTGER4 P35408 3/20 0.39
PTGER3 P43115 1/20 0.38
CYP19A1 P11511 1/20 0.38
TSHR P16473 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
POLB P06746 2/20 0.37
TACR1 P25103 4/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
CDC7 O00311 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638478 0.94 ADORA3 (0.41) ALDH1A1GAAADORA3PTGER4PTGER3
SCHEMBL4637770 0.94 ADORA3 (0.46) ALDH1A1GAAADORA3PTGER4AKR1C3
SCHEMBL4637820 0.88 GAA (0.40) ALDH1A1GAAADORA3PTGER4CYP19A1
SCHEMBL4638051 0.88 ALDH1A1 (0.39) ALDH1A1GAAADORA3PTGER4PTGER3
SCHEMBL4638558 0.87 ALDH1A1 (0.42) ALDH1A1GAAADORA3PTGER4PTGER3
SCHEMBL4637826 0.82 ALDH1A1 (0.47) ALDH1A1GAAADORA3PTGER4CYP19A1
SCHEMBL4637811 0.81 GRM2 (0.36) ALDH1A1GAAADORA3PTGER4PTGER3
SCHEMBL4638520 0.80 ALDH1A1 (0.44) ALDH1A1GAACYP19A1TSHRAKR1C3
SCHEMBL4638481 0.79 IDH1 (0.44) GAAGPBAR1TACR1
SCHEMBL4637948 0.79 RORB (0.36) ADORA3GPBAR1AKR1C3AKR1C2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed