SCHEMBL4637770

SCHEMBL4637770

O=C(C#Cc1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.46
PTGER4 P35408 3/20 0.42
POLB P06746 2/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
LRRK2 Q5S007 1/20 0.39
ADCY1 Q08828 1/20 0.38
VNN1 O95497 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637822 0.94 ALDH1A1 (0.43) ADORA3PTGER4POLBAKR1C3AKR1C2
SCHEMBL4638478 0.89 ADORA3 (0.41) ADORA3PTGER4POLBAKR1C3AKR1C2
SCHEMBL4637820 0.85 GAA (0.40) ADORA3PTGER4POLBAKR1C3AKR1C2
SCHEMBL4638051 0.84 ALDH1A1 (0.39) ADORA3PTGER4AKR1C3AKR1C2ALDH1A1
SCHEMBL4638558 0.83 ALDH1A1 (0.42) ADORA3PTGER4POLBAKR1C3AKR1C2
SCHEMBL4637775 0.81 POLB (0.45) ADORA3PTGER4POLBAKR1C3AKR1C2
SCHEMBL4637826 0.79 ALDH1A1 (0.47) ADORA3PTGER4POLBAKR1C3AKR1C2
SCHEMBL4637811 0.78 GRM2 (0.36) ADORA3PTGER4AKR1C3AKR1C2ALDH1A1
SCHEMBL4638520 0.77 ALDH1A1 (0.44) POLBAKR1C3AKR1C2ALDH1A1GAA
SCHEMBL4638481 0.76 IDH1 (0.44) GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed