SCHEMBL4638841

SCHEMBL4638841

CC(C)(C)[Si](C)(C)OCc1onc(-c2c(F)cccc2F)c1C(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1N1CCOCC1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
POLB P06746 2/20 0.33
TSHR P16473 1/20 0.33
KCNH2 Q12809 3/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
USP2 O75604 2/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 3/20 0.32
CETP P11597 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
LMNA P02545 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639398 0.93 KMT2A (0.37) TACR1MEN1KMT2APOLBTSHR
SCHEMBL4639495 0.87 TACR1 (0.31) TACR1MEN1KMT2APOLBTSHR
SCHEMBL4637842 0.87 TACR1 (0.36) TACR1MEN1KMT2APOLBTSHR
SCHEMBL4638040 0.85 ALDH1A1 (0.31) TACR1L3MBTL1ALDH1A1
SCHEMBL4638555 0.85 CNR1 (0.32) L3MBTL1ALDH1A1
SCHEMBL4638545 0.82 ALDH1A1 (0.38) TACR1MEN1KMT2APOLBTSHR
SCHEMBL4637966 0.80 KMT2A (0.41) TACR1KMT2APOLBMAPTSMN1; SMN2
SCHEMBL4639400 0.76 NR1H4 (0.37) KMT2ATSHRL3MBTL1KDM4EALDH1A1
SCHEMBL4637694 0.76 EPAS1 (0.39) TACR1MEN1KMT2APOLBTSHR
SCHEMBL4637876 0.76 EPAS1 (0.39) TACR1MEN1KMT2APOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed