SCHEMBL4639495

SCHEMBL4639495

CC(C)(C)[Si](C)(C)OCc1onc(-c2cccnc2Cl)c1C(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1N1CCOCC1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.31
ALDH1A1 P00352 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
TSHR P16473 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639459 0.89 TACR1 (0.34) TACR1TP53MAPT
SCHEMBL4638555 0.89 CNR1 (0.32) ALDH1A1TDP1L3MBTL1
SCHEMBL4638040 0.89 ALDH1A1 (0.31) TACR1ALDH1A1TDP1L3MBTL1
SCHEMBL4639398 0.89 KMT2A (0.37) TACR1ALDH1A1TDP1L3MBTL1TP53
SCHEMBL4638841 0.87 TACR1 (0.34) TACR1ALDH1A1L3MBTL1TP53MAPT
SCHEMBL4638545 0.86 ALDH1A1 (0.38) TACR1ALDH1A1TDP1L3MBTL1MAPT
SCHEMBL4637876 0.81 EPAS1 (0.39) TACR1ALDH1A1TDP1L3MBTL1MAPT
SCHEMBL4637694 0.81 EPAS1 (0.39) TACR1ALDH1A1TDP1L3MBTL1MAPT
SCHEMBL4638045 0.80 EPAS1 (0.39) TACR1ALDH1A1TDP1L3MBTL1MAPT
SCHEMBL4637747 0.80 EPAS1 (0.38) TACR1ALDH1A1TP53MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed